Detailed Scientific Program

Day by Day Program

Instruction for Oral Session Speakers

The session rooms are provided with one LCD projector for laptop computer presentation. Laptop computers are loaded with “power Point 2003” with 2007 compatibility so you can run 2007 files but cannot edit these files. Each session room will have this as will the Fortune Bay room which will be available for delegates to use prior to their presentation and throughout the conference. Staff will be available to assist on request. Plenary Lectures will be 1 hour in length while Invited Lectures will last 30 minutes. Oral Contributions will be strictly limited to 20 minutes each. A bell will ring 3 minutes before the end of each presentation (oral presentation), 5 minutes before the end (invited talks), and 10 minutes and 5 minutes before the end for plenary presentations.

Instruction for Poster Presentation

Poster boards will accommodate posters 6’ wide x 3’ high. Posters can be attached to the boards using double sided Velcro. Author(s) are asked to place their materials on the assigned board prior to the sessions, beginning at 12:30, and remove them at the end of the poster session. The poster presentations will be held as indicated below: Poster Session PO-O1 to PO-52 Monday August 3, 5:00 pm – 6:30 pm Poster Session PO-53 to PO-109 Tuesday August 4, 5:00 pm – 6:30 pm

LECTURE & POSTER PROGRAM

Monday August 3, 2009

Main Session (Salon A)

PL-1 9:00-10:00
Adventures in heterocyclic compound synthesis
Steven V. Ley

IL-1 10:00-10:30
Novel Sphingosine 1-Phosphate Receptor Agonists:
Asymmetric Synthesis of Thiophene and Pyrrole Analogues
Takahide Nishi

PL-2 11:00-12:00
Development of a facile synthetic strategy for bioactive alkaloids possessing a spirocyclic ring system
Toshio Honda

IL–2 12:00-12:30
Making and Breaking Heterocyclic Rings via Metal Catalyzed Reactions
Mark Lautens

IL-3 1:30-2:00
Synthesis of Heterocycles via Alkoxyallenes
Hans-Ulrich Reissig

OL-1 2:00-2:20
Fused/Isolated Heterocyclic of Pyrrole, β-Lactam, Thiazolidine and Triazine Derivatives.
H.A. Soleiman

OL-2 2:20-2:40
ß-Dimethylamino-a,ß-Didehydro-a-Amino acid derivatives and related enaminones in the synthesis. Versatile reagents for preparation of various heterocyclic systems
Branko Stanovnik, Uroš Uršic, and Jurij Svete

OL-3 2:40-3:00
Heterocycle Synthesis Triggered by Oxygen-Nitrogen Bond Cleavage
Okiko Miyata, Partha P. Mukhopadhyay, Takeaki Naito

IL-4 3:30-4:00
Enantioselective Desymmetrization of 2-Substituted Glycerols and its Synthetic Application to Azithromycin
Hyoung Cheul Kim, Byunghyuk Jung and Sung Ho Kang

OL-4 4:00-4:20
Total Synthesis of Norzoanthamine
Daisuke Yamashita, Yoshihisa Murata, Atsuo Nakazaki, and Susumu Kobayashi

OL-5 4:20-4:40
The total synthesis of hyacinthacine B3 and putative hyacinthacine B7
Stephen G. Pyne

OL-6 4:40-5:00
Application of Dipolar Cycloadditions and C-2 Alkylation of Indoles Involving Donor-Acceptor Cyclopropanes: Synthesis of (±)-Quebrachamine and Tetrahydroisoquinocarbazoles.
Barbora Bajtos and Brian L. Pagenkopf

Session 1 (Salon C)

IL-5 1:30-2:00
Synthesis of bipyridine N,N’-dioxides and their application enantioselective reactions
Martin Kotora
OL-7 2:00-2:20
New and Efficient Route for Synthesizing Tetrahydro-benzo-4H-[1,3]-oxazines using TCS/ ZnCl2 Reagent Mixture.
Wahid M. Basyouni , Khairy A.M. El-Bayouki , Ezzat M. Kandee, Doria S. Badawy, Ebrahim Abdel-Galil and Tamer K.A. Khattab.

OL-8 2:20-2:40
Heterocyclic Synthesis through Asymmetric aza-Baylis-Hillman Equivalent Reaction
Akio Kamimura and Shingo Ishikawa

OL-9 2:40-3:00
Non-traditional synthesis of novel heterocyclic compounds
Antonin Klasek, and Antonin Lycka

OL-10 3:30-3:50
Design, Synthesis and Pharmacological Evaluation of New Nonsteroidal Anti-inflammatory Derived from 3-Aminobenzo-thieno[2,3-d]pyrimidines
H. N. Hafez and A. B. A. El-Gazzar

OL-11 3:50-4:10
An intramolecular Wolff rearrangement toward β-lactams
Yvette M. Vaske and Joseph P. Konopelski

OL-12 4:10-4:30
Facile Synthesis of Novel Imidazo[5,1-b][1,3,4]oxadiazoles and their Imidazo-thiadiazole Analogues
Nandini Patel, Brian Samas, Jacob B. Schwarz, and Tuan P. Tran

OL-13 4:30-4:50
Synthesis of 5-membered heterocycles by SmI2-promoted intramolecular coupling reaction of alkynes with a,ß –unsaturated ester
Kazunori Takahashi and Toshio Honda

Session 2 (Salon D)

IL-6 1:30-2:00
Enantioselective Reactions Catalyzed by Chiral Pyridine 2,6-Bis(5',5'-diphenyloxazoline)-Cu(II) Complexes
Vinod K. Singh

OL-14 2:00-2:20
Synthesis of indoles, N-alkoxyindoles, and quinolines from reductive N-heteroannulation of 2-nitrostyrene derivatives
Björn C. G. Söderberg and Serge R. Banini

OL-15 2:20-2:40
New Zwitterionic Pyridine Derivatives as Valuable Starting Materials for Rearrangements
György Hajos and Roberta Palko

OL-16 2:40-3:00
Planar-chiral pyridinophanes as new synthetic tools for enantioselectivecyclopropanation reactions
Nobuhiro Kanomata, Ryo Sakaguchi, Kiichiro Nishimura, Hironobu Kubota, and Kazuki Kimura

OL-17 3:30-3:50
Conversion of Isothiazoles into Pyrazoles with Hydrazine
Herakildia A. Ioannidou, Panayiotis A. Koutenis

OL-18 3:50-4:10
Synthesis of Axially Chiral a,ß -Unsaturated Amidines via Stereoselective Cycloreversion of 2-Aminoazetines
Kiyosei Takasu, Naoya Shindoh, and Yoshiji Takemoto

OL-19 4:10-4:30
Scaffold Decoration of Heterocycles With Embedded Thioamide Motifs Applying Desulfitative Carbon-Carbon Cross-Coupling Chemistry
Hana Prokopcová, Nuzhat Arshad, and C. Oliver Kappe

OL-20 4:30-4:50
Photocycloaddition and Pulse Radiolytic Studies on some Hetero-1,4-benzoquinones
R.T.Pardasani, Ignatious Abraham, Praveen Khatri and T.Mukherjee

Posters (Salon B) 5:00-6:30

PO-1
Some Observations on the Base-Catalyzed Cyclocondensation of 2,6-Dihalobenzaldehydes, Ethyl Cyanoacetate, and Thiourea
Mohamed A. Al-Omar, Abdul-Rahman M. Al-Obaid, Nasser R. El-Brollosy, and Ali A. El-Emam

PO-2
PEG-SO3H as an eco-friendly catalyst for the efficient synthesis of 1,8-dioxo-octahydroxanthenes and 1,8-dioxo-decahydroacridines in different conditions
Alireza Hasaninejad, Mohsen Shekouhy

PO-3
Chemical Confirmation of the Structure of a Biologically Derived Carcinogen, 9-(4’-Aminophenyl)-9H-pyrido[3,4-b]indole. An Authentic Synthesis of 9-(4’-Nitrophenyl)-9Hpyrido[3,4-b]indole as the Relay Compound.
Yasuoki Murakami, Nobuyuki Imai, Tsuyoshi Miura, Takashi Sugimura, Keiji Wakabayashi,Yukari Totsuka, Noriyasu Hada, Yuusaku Yokoyama, Hideharu Suzuki, and Katsuyoshi Mitsunaga

PO-4
Convenient synthesis of 1,2,4-triazole-3-thiones and heterocyclic systems containing 1,2,4-triazole ring
Mitsuo Kodomari, Shota Kanno, and Tadashi Aoyama

PO-5
Facile synthesis of 3-substituted pyrazoles and indazoles using [3+2]cycloaddition reactions of 2-diazo-2-(trimethylsilyl)ethanols
Yoshiyuki Hari, Ryosuke Sone and Toyohiko Aoyama

PO-6
Chiral Lewis acid catalyzed asymmetric cycloaddition reactions of cyclic ylides generated from diazocarbonyl compounds
Hiroyuki Suga, Satoshi Higuchi, Motoo Ohtsuka, Shingo Yasumura, and Ayano Inaba

PO-7
A Convenient Synthesis Of bis (indole) alkanes by nobium ( V) chloride
Majid M. Heravi, Fatemeh.Nahavandi

PO-8
Synthesis of 2-(N-alkylamino)thiazoles and N-thiazolo-1,3-oxathiol-2-imines using supported reagents
Tadashi Aoyama, Sumiko Murata, Izumi Arai, Toshio Takido, and Mitsuo Kodomari

PO-9
Synthesis of novel 2-thioxo-1´H-spiro[imidazoline-5´-indole]-2,2´-diones.
Antonín Klásek, Vladimír Mrkvicka, Antonín Lycka, Ivan Mikšík, and Aleš Ružicka

PO-10
High Pressure and Microwave-mediated Synthesis of 2-Pyridones by Hilbert-Johnson Reaction
Hirokazu Iida, Yuka Nagashima, Kouta Joho, Tatsuya Moromizato, Seisuke Mimori, Yasuoki Murakami, Kiyoshi Matsumoto, and Hiroshi Hamana

PO-11
Facile preparation of a highly functionalized tetrahydropyran by catalytic hydrogenation of an oxazoline
Dusan Hesek, Mijoon Lee, Takao Yamaguchi and Shahriar Mobashery

PO-12
Microwave-Assisted Synthesis of 2-Pyridones and Their Nucleoside Analogues
Ibrahim M. Abdou and Alaa A. Salem

PO-13
One-pot synthesis of N,N’-dialkyl-7,7’-diazaindigos from N-alkyl-7-azaindoles
Jiro Tatsugi, Maki Miura, and Kouta Maedera

PO-14
Bronsted acidic ionic liquid as an efficient catalyst for synthesis of aryl-14H-dibenzo [a.j] xanthenes under solvent-free conditions
Abdol R. Hajipour and Arnold E. Ruoho

PO-15
Synthesis and characteristics of a novel artificial nucleoside bearing a 6-oxa-2,3-dithiabicyclo[3.2.1]octane skeleton
Takeshi Baba, Tetsuya Kodama, Takeshi Imanishi, Satoshi Obika

PO-16
Practical synthesis of axially chiral amino acid through efficient construction of aza[5]helicenes
Takumi Furuta, Junya Yamamoto, Yuki Kitamura, Ayano Hashimoto, Hyuma Masu, Isao Azumaya, Toshiyuki Kan and Takeo Kawabata

PO-17
An efficient microwave assisted synthesis of 1,4-benzothiazine and 1,5-benzodiazepine
Ola Ghoneim

PO-18
Thermal Isomerization of Benzylselenocyanate. Flash Vacuum Pyrolysis as Alternative Synthesis of Building Blocks towards Selenoheterocycles
Noelia M. Ceballos and E. Laura. Moyano

PO-19
Syntheses of heterocyclic compounds derived from new type of a-trifluoromethyl-ß-aminoalcohols
Emilia Obijalska, and Grzegorz Mloston

PO-20
Synthesis of 2,3-dihydro-imidazo[2,1-b]thiazole derivatives via cyclizationof 1-allyl-4,5-disubstituted-imidazole-2-thiones
Marcin Jasinski, Grzegorz Mloston

PO-21
Regioselective synthesis of 3-aroyl imidazo[1,2-a]pyridines
Héctor Salgado-Zamora, Omar Gómez, Cuauhtémoc Pérez and María Elena Campos

PO-22
Progress Toward the Synthesis of Complex Fused-Ring Mesoionic Heterocycles, Including Microwave Assistance
Douglas Armstrong

PO-23
Synthesis of novel molecules with both Biginelli and Diindolylmethane moieties.
José Guillermo Penieres Carrillo, Noelia Ceballos, Elizabeth Laura Moyano, Eugenia Guadalupe Ramírez Guido, José Ernesto Valdez Rojas

PO-24
Study of a new methodology for the synthesis of alpha-ketochalcogenoamides
José Ernesto Valdez Rojas, José Guillermo Penieres Carrillo*, Josefina Juárez Reséndiz, Guadalupe García González.

PO-25
Regioselective synthesis of unsubstituted basic skeletons of heterocycles containing nitrogen neighboring an aromatic ring by the reductive ring expansion reaction using diisobutylaluminum hydride (DIBAH)
Hidetsura Cho, Yusuke Iwama, Kenji Sugimoto, Seiji Mori, Eunsang Kwon, and Hidetoshi Tokuyama

PO-26
Tandem reaction to naphto[1,8-bc]furan ring via intramolecular Diels-Alder reaction
Noriyuki Hatae, Tatsunori Iwamura

PO-27
Reaction Of 1,10-Diaza-18-Crown-6 with Allenylphosphonates
Narkis Khusainova, Sergey Rybakov, Damir Safin, Mikhail Khusainov, Aygul Khakimullina, Rafael Cherkasov

PO-28
Reaction Of 2-H-1,2,3-Diazaphosphole with 1,2-Ethanedithiol
Narkis Khusainova, Olga Mostovaya, Mikhail Khusainov, Svetlana Slivko, Rafael Cherkasov

PO-29
Reaction of 3-amino-1H,3H-quinoline-2,4-diones with thiourea and potassium thiocyanate
Vladimír Mrkvicka, Antonín Lycka, Ondrej Rudolf, Antonín Klásek

PO-30
Reactions of Thiazazulanone and Thiazazulathione with Dimethyl Malonate Derivatives
Ohki Sato, Nobuhiro Ando, Tatsuro Toma, Hiroshi Onuma and Juzo Nakayama

PO-31
Substituent effects on rope-skipping isomerization of planar-chiral parapyridinophanes
Yasuyuki Ueda, Kazuki Kimura, Nobuhiro Kanomata

PO-32
Guanidinyl Pyrrolidines as Bifunctional Organocatalysts for Asymmetric Conjugate Addition Reactions
Rajinikanth Lingampally and Sunil V. Pansare

PO-33
New hydrazides of imidazolecarboxylic acids and their exploitation for the syntheses of polyheterocyclic compounds
Adam Marek Pieczonka, and Grzegorz Mloston

PO-34
Recent Developments on the 1,2,3-Dithiazole to Isothiazole Conversion
Heraklidia A. Ioannidou, Andreas S. Kalogirou and Panayiotis A. Koutentis

PO-35
The reaction of 3-nitroimidazo[1,2-a]pyridine-2-carbonitrile with nucleophiles
Jorge Hernández, Héctor Salgado-Zamora, Humberto Cervantes, Lucina Arias and Ma. Elena Campos

PO-36
An intramolecular hydrogen bridge involved in conformational preference and in a plausible explanation of the peri effect in 3-substituted imidazo[1,2-a]pyridines
Héctor Salgado-Zamora, Manuel Velázquez, Daniel Mejía-Rodríguez, Hugo Jiménez, Maria Elena Campos and Rogelio Jiménez.

PO-37
Generation and Characterisation of the Elusive 1,4-Oxazine
R. Alan Aitken, Kati M. Aitken, Philip G. Carruthers and Marc-Alexandre Jean

PO-38
Versatile Thermal Behaviour of Spiro 1,3-Dioxolan-4-ones Leading to New Heterocyclic Syntheses
R. Alan Aitken, Alan R. Henderson and Lynn A. Power

PO-39
Synthesis and Anti-Tumour Activity of [1,2-a] Alicyclic Ring Fused Benzimidazolequinones Containing Reactive Aziridine Rings
Karen Fahey, Liz O’Donovan, Michael P. Carty and Fawaz Aldabbagh

PO-40
Synthesis, Antimicrobial, and Anti-inflammatory Activities of Novel 3-(1-Adamantyl)-1-arylideneamino-5-mercapto-1,2,4-triazoles and Related Derivatives
Mohamed A. Al-Omar, Ebtehal S. Al-Abdullah, Ihsan A. Shehata, and Ali A. El-Emam

PO-41
Synthetic studies toward the novel peptide nucleic acid monomers by application of 4-hydroxyproline as backbone synthon
Akiko Watanabe, Naotoshi Kiyota, Tatsunori Miyagoe, Atsushi Toyao, Tetsuo Yamasaki, Masanori Sakamoto, and Masami Otsuka

PO-42
Design and syntheses of benzoquinolines as potential topoisomerase inhibitors
Abeer Ahmed, and Mohsen Daneshtalab

PO-43
Design, Syntheses & Biological Evaluation of Thieno[2,3-b]quinolones as Topoisomerase poisons
Ranjith Garlapati, and Mohsen Daneshtalab

PO-44
Microwave assisted synthesis, X-Ray analysis, DFT study and antioxidant activity of two novel 1,4-dihydropyridine derivatives of 4-hydroxycoumarin
Stefan Dochev, Ilia Manolov, Vessela Kancheva, Pascal Retailleau, Anita Penkova

PO-45
Synthesis and evaluation of 2-arylbenzimidazole derivatives against Chlamydia pneumoniae
Leena Keurulainen, Olli Salin, Antti Siiskonen, Heikki Vuorela, Pia Vuorela, Jari Yli-Kauhaluoma, Paula Kiuru

PO-46
Design & synthesis of 5-(4-Substituted benzyl)-2-methylsulfonyl-1,3,4-oxadiazoles: a novel class of cyclooxyenase-2 inhibitors
Bahar Mokarami

PO-47
Synthesis and screening of a 16,000 compound library of stereochemically diverse macrolactams
Maurice duPont Lee IV, Eamon Comer, Sivaraman Dandapani, Jason Lowe, Haibo Liu, Carol Mulrooney, Byung-Chul Suh, Damian Young, Lisa Marcaurelle

PO-48
Diindolylmethanes as apoptosis inductors in L5178Y cells
José Guillermo Penieres Carrillo, Benjamín Velasco Bejarano, Luvia Enid Sánchez Torres, José Guadalupe García Estrada, René Miranda Ruvalcaba, Cecilio Álvarez Toledano

PO-49
Synthesis of New MMP Inhibitors and Evaluation of Their MMP-Inhibitory Activity
Naoki Tanaka, Kazuya Emi, Satoshi Onoe, Masahiro Fukumori, Akiko Tsukamoto, Yoshito Zamami, Chie Ohtsuka, Seiji Tsuboi, and Kenji Sasaki

PO-50
Water Soluble Chitosan derivatives as antimicrobial agents
Ahmad Reza Ghanbarpour, Pouneh Ebrahimi, Fereshteh Pourmorad

PO-51
Prediction of solubility of new water- soluble chitosan derivatives
Fereshteh Pourmorad, Pouneh Ebrahimi, Ahmad Reza Ghanbarpour, Mohammad Ali Ebrahimzadeh, Soheila Honary

PO-52
Studies toward the synthesis of tetrathiacalix[4]arene(amido)crowns
Suneel Pratap Singh and Har Mohindra Chawla

Tuesday August 4, 2009

Main Session (Salon A)

PL-3 9:00-10:00
Proximity-Assisted Stereocontrolled Cycloaddition Reactions of Acetals
Stephen Hanessian

SNIECKPOSIUM:

a tribute to Professor Victor Snieckus

“Focuc on Heterocycles in Organic Synthesis Today and Tomorrow”

PL-4-S 10:00-11:00
Cooperativity in Catalysis: A Novel Method for Enantioselective Transformations with Complex Substrates
Mukund P. Sibi

IL-7-S 11:30-12 :00
Asymmetric Synthesis: The Complex Induced Proximity Effect and Dynamic Thermodynamic Resolution
Peter Beak, Suk Joong Lee, & Yong Sun Park

IL-8-S 12:00-12:30
Design, Synthesis and Biological Evaluation of Novel TNF-a Converting Enzyme(TACE) Inhibitors
M.Arshad Siddiqui

IL-9-S 1:30-2:00
Catalytic Organometallic Carbon-Heteroatom Bond Formation
John F. Hartwig, Kenneth L. Rinehart Jr.

IL-10-S 2:00-2:30
Overview of recent Chemoenzymatic Total Syntheses of Natural and Unnatural Products: Codeine, Balanol, Pancratistatin, & Tamiflu
Tomas Hudlicky

IL-11-S 2:30-3:00
Toward A Fundamental Understanding of Asymmetric Phase Transfer Catalysis
Scott E. Denmark

Chaired by Professor Tomas Hudlicky
OL-21-S 3:30-3:50
Unexpected One-pot Sequential Halogen Dance-Anionic Ortho Fries Rearrangement of Iodo O-Aryl Carbamates
Ricarda E. Miller, Ulrich Groth, Victor Snieckus

OL-22-S 3:50-4:10
Iridium(I) Complexes Bearing Chiral Phenanthroline-Derived Benzimidazolylidenes: Synthetic, Structural & Catalytic Studies
Costa Metallinos and Xiangdong Du

OL-23-S 4:10-4:30
The Synthesis of Velloziolide
J. R. Green & A. A. Tjeng

OL-24-S 4:30-4:50
Synthesis of Higher Carbohydrates On Dioxanone Scaffold
Marek Majewski, Nagarjuna Palyam & Izabella Niewezas

Session 1 (Salon C)

OL-25-S 3:30-3:50
Synthesis of 1-Methylphenanthrene Metabolites by Directed Metalation Strategies
Kare B. Jorgensen, Toni Rantanen, Thilo Dorfler and Victor Snieckus

OL-26-S 3:50-4:10
Organosilicon reagents in Palladium Catalysed Cross Coupling Reactions with Aryl and Heteroaryl Halides
H. F. Sore, C.M. Boehner, D.R.Spring, S.J.K. MacDonald

OL-27-S 4:10-4:30
A Zinc(II) Catalyzed Synthesis of Piperidines from Propargyl Amines and Donor-Acceptor Cyclopropanes
Terry P.Lebold, Andrew B. Leduc, Michael A. Kerr

OL-28-S 4:30-4:50
A Roundabout ortho Metallation of Benzyl Alkynyl Sulfones for Eventual Cyclization to Benzothiopyran Dioxides
Adrian L. Schwan and Md. Selim Hossain

Session 2 (Salon D)

OL-29 3:30-3:50
New S-nucleoside Analogues Derived from Thieno[2,3-d] Pyrimidines As Potential Analgesic and Anti-inflammatory Activities.
A. B. A. El-Gazzar, H.N.Hafez, G.A.M. Nawwar

OL-30 3:50-4:10
Studies Towards The Synthesis Of Homocytisine & Investigations Into the Scope of Intramolecular 1,6-additions
Claire Haseler, Timothy Gallagher

OL-31 4:10-4:30
Push-Pull Substituted Alkinyl Thiophenes- Metal-Free Molecules With Small Homo-Lumo Gaps
Eva-Janina Vogt, Viktor Zapol’ skii and Dieter E. Kaufmann

OL-32 4:30-4:50
Synthesis and Reactions of 1-Azetines, other Cyclic Imines, ß- sultams and ?-sultams
Arnaud Pitard, M.Hyas Qamar and Karl Hemming

Posters (Salon B) 5:00-6:30

PO-53-S
Investigating RebC-Mediated Chemoselective Oxidation During Rebeccamycin Biosynthesis
Katherine A.Groom, V.Snieckus, D.Zechel

PO-54-S
Palladium Catalyzed Direct Heck Coupling At C-5 Of Imidazo[1,5-a]Pyrazines
Jian-Xin Wang, J.Adam McCubbin, Meizhong Jin, Andrew P.Crew, Radoslaw S. Laufer, Yunyu Mao, Mark J. Mulvihill, Jonathan Board, & Victor Snieckus

PO-55-S
Studies Towards the Total Synthesis of Isoprekinamycin: A New Metallation Route to 2-Naphthols From Coumarin-2-ones
Jignesh J. Patel, Manlio Alessi, Emilie David & Victor Snieckus

PO-56-S
Synthesis of Regioisomeric Aryl Boronates Via Complementary Methodologies
Hurst, T. Macklin, T. Hartmann, E. Kugel, W. Parisienne-La Salle, J.-C., Becker, M., Schneider, C., Marder, T., Snieckus, V.

PO-57-S
Reduction of Tertiary Amides To Aldehydes By in situ Generated Schwartz Reagent [Cp2Zr(H)Cl]. Link to the directed ortho Metalation (DoM) Reaction
Yigang Zhao, Justin Morin, & Victor Snieckus

PO-58-S
Towards the Synthesis of Lysergic Acid Via a Directed ortho Metalation(DoM) Strategy
Yigang Zhao, Andrew Larkin, & Victor Snieckus

PO-59-S
Synthesis of A New Liquid Crystal (LC) Material with Phenanthrene Core by A Combined Metalation-Cross Coupling Strategy
Wei Gan, Victor Snieckus, Robert Lemieux

PO-60-S
Synthesis of New Troger’s Base Derivatives
Josefine Karlsson, Erhad Ascic, Victor Snieckus, Kenneth Warnmark, Michael Harmata

PO-61-S
A Novel Base Induced Cyclization of Benzyl Alkoxyl Sulfones
M Selim Hossain and Adrian L. Schwan

PO-62
Selenium-Containing Heterocycles 2 A Straightforward Double Intramolecular Cyclization of Dibenzyl Diselenols into an Ethynyl Group
Haruki Sashida, Akemi Nakayama, and Mamoru Kaname

P0-63
Selenium Containing Heterocycles 1One-Pot Synthesis of (Z)-1-Methylidenebenzo[c]selenophenes From o-Ethynylbomobenzenes and Isoselenocyanate
Mamoru Kaname and Haruki Sashida

PO-64
Domino Process of Iodocyclization and Diels-Alder Reaction for the Construction of Bridgehead-Spiro Heterocycles Takashi Okitsu, Daisuke Nakazawa, and Akimori Wada

PO-65
The Synthesis of 6-alkylidene Substituted 1,1-Dioxopenicillanates
Irina Potorocina, Maksim Vorona, Grigory Veinbarg, Irina Shestakova, Sergi Belyakov, Edmunds Lukevics

PO-66
Highly Efficient Synthesis of 2,5- or 2,6- Bridged Pyridine: Intramolecular [4+2] Cycloaddition of Bis(Acylketene) Followed By Ring Transformation
Masayuki Sato, Kie Suwa, Katsuya Fusazaki, Yasuko Morie, Kiyoshi Ikeda, Yumiko Suzuki, Ken-ichi Iwamoto

PO-67
New Dihydro-TTF-Quinone Donor-Acceptor Compounds For Attachment To Metal Surfaces
Kati M. Aitken, R. Alan Aitken, Stephen J. Costello & Neil J. Wilson

PO-68
Intramolecular Cross Coupling Of gem-dibromo-Olefins: A Mild Approach to Halogenated Benzofused Heterocycles
Stephen G. Newman, Valentina Aureggi, Christopher S. Bryan, Mark Lautens

PO-69
Highly Efficient Macrolactonization Method Via ethoxyvinyl Ester
Yusuke Ohba, Mayuko Takatsuji, Kenji Nakahara, Hiromichi Fujioka, and Yasuyuki Kita

PO-70
New Generation of Recyclable Hypervalent Iodine Reagents And Catalysts
Toshifumi Dohi, Akinobu Maruyama, Naohiko Washimi, Naoko Takenaga, Hiromichi Fujioka, & and Yasuyuki Kita

PO-71
Design of New Hypervalnet Iodine(III) Reagents And Their Application in Assymetric Phenolic Oxidations
Naoko Takenaga, Akinobu Maruyama, Daishi Kato, Hiromichi Fujioka, Toshifumi Dohi, and Yasuyuki Kita

PO-72
Metal Free Biaryl Coupling Reactions Of Heteroaromatic Compounds Using Hypervalent Iodine(III) Reagent
Koji Morimoto, Motoki Ito, Chieko Ogawa, Hiromichi Fujioka, Toshifumi Dohi, and Yasuyuki Kita

PO-73
Organoiodine(III)-Induced Oxidative Cross-Biaryl-Coupling Via Selective Single Electron-Transfer Process
Motoki Ito, Nobutaka Yamaoka, Koji Morimoto, Hiromichi Fujioka, Toshifumi Dohi, and Yasuyuki Kita

PO-74
Concise Synthesis of Benzocoumarins And C2-Symmetric Pyrenophanes
Penchal Reddy Nandaluru, Graham J. Bodwell

PO-75
[4+2] Cycloaddition of 1-Aza- and 1,2,4-Triaza-1,3-dienesWith Diphenylketene
Masanori Sakamoto, Tatsuya Nakai, Kyoko Fukutomi, Hiroaki Yanagisawa, Tomomi Kawasaki

PO-76
Synthesis of Chiral Cyclic Amines Via Diastereoselective Addition of Grignard Reagents to Imines and Oxazolidines and Ring-Closing Metathesis
Kimio Higashiyama, Ryuji Ogusa, Takayasu Yamauchi, and Shigeru Sasaki

PO-77
Dual Activation of carbonyl Groups with Bronsted and Lewis Acids: Proof of Principle Experiments
Seiji Hata and Mukund P. Sibi

PO-78
Synthesis of 2,3-Dibromoindoles by Decarboxylative Bromination of Indole-2,3-Dicarboxylic Acids
Yasuyoshi Miki, Misako Umemoto, Chiaki Ota, Masashi Doshita, Hiroki Tanaka, Hideaki Umemoto, Hiromi Hamamoto

PO-79
Catalytic Aziridination of Electron-Deficient Olefins Using N-Haloamides and Its Application to Asymmetric Synthesis
Satoshi Minakata, Yuta Murakami

PO-80
Solid Base Effects On Lewis Acid-Catalyzed Stereoselective Nitrile Oxide Cycloaddition Reactions
Hidetoshi Yamamoto, Yuji Ikenaga, Maki Samitsu, Masahiro Komeda, Saori Hayashi, Michinori Sumimoto, and Kenji Hori

PO-81
Influence of Some Heterocyclic Lewis Bases on Liquid Crystalline And Luminiscence Properties of Their tris(ß-diketonates) Adducts with Lanthanides
Yury Galyametdinov, Andrey Knyazev, Vagif Dzhabarov, Elena Molostova

PO-82
Catalytic Cyclopropanation Reactions Via Pyridinium Ylides Generated From Copper Carbenoid Complexes
Hiroko Tanaka and Nobuhiro Kanomata

PO-83
Fluoride-Free Cross-Coupling Using Disiloxanes
C.M.Boehner, H.F.Sore, D.R. spring, D. Norton

PO-84
Synthesis of Novel Luminiscent 5-Hydroxythiazoles
E.Tauscher, K. Stippich, D. Weib, R. Menzel, R.Beckert

PO-85
A New Synthetic Route To The 1-Oxygenated Carbazole Alkaloids, Mukonine and Clausine E (Clauzoline I)
Satoshi Hibino, Shigeo Tohyama, Shuhei Azuma, Haruto Fujioka, and Tominari Choshi

PO-86
Novel Synthesis of The 2-Aza-anthraquinone Alkaloid, Scorpinone, Based on Two Microwave Assisted Pericyclic Reactions
Tominari Choshi, Teppei Kumemura, Junko Nobuhiro, and Satoshi Hibino

PO-87
A New Synthesis of the Benzo[c]phenanthridines, Nornitidine, Noravicine, And Isodecarine Based On A Microwace-Assisted Electrocyclic reaction of the Aza 6p- Electron System
Shuhei Azuma, Kakujiro Kohno, Tominari Choshi, Junko Nobuhiro, and S.Hibino

PO-88
Progress Towards The Synthesis Of Cyclocinamide A & B
Jessica M Garcia, Stephanie S. Curzon, and Joseph P. Konopelski

PO-89
Synthesis of Polyfunctionalized Pyridines Via Hetero Diels-Alder Reaction Of the Isotellurazoles with Acetylenic Dienophiles & Their Application to the Construction of Fused Pyridine Alkaloid Skeletons
Kazuaki Shimada, Yukichi Takata, Yu Osaki, and Satoshi Oawa

PO-90
Synthetic Study Of Azinomycin A Via a 3,4-Epoxypiperidine Structure
Yuji Kawada, Takao Yamaguchi, Kazuyuki Miyashita, Takeshi, Imanishi, and Satoshi Obika

PO-91
Enantioselective Total Synthesis Of Some Bisbenzyltetrahydoisoquinoline Alkaloids Ahmed L. Zein and Paris E.Georghiou

PO-92
Cobalt Catalyzed [2+2+2] Cycloadditions Of Diyne-Cyanohydrins To Natural Product Analogs
Anja Meissner and Ulrich Groth

PO-93
Total Synthesis of Himeic Acid A & B
Takeshi Shimizu, Kohei Matsushige, and Mikiko Sodeoka

PO-94
A New Access To Azepinoindole Alkaloids Through Base- Promoted Pictet-Spengler Reaction
Koji Yamada, Tomohiro Haruyama, Yuuichi Namerikawa, and Minoru Ishikura

PO-95
Stereoselective Synthesis of 2,5-Disubstituted Tetrahydofurans Using 8-Oxabicycli[3.2.1] Octane Platform: Building Blocks For Natural Products
Arun A. Yadav, Donald F. Weaver, Girish K. Trivedi, and Manikrao M. Salunkhe

PO-96
Synthesis of ?-Valerolactones As The Tea Catechin Metabolites
Masahiro Hamada, Sousuke Nakano, Takao Kishimoto, and Noriyuki Nakajima

PO-97
A Cyclic Pentapeptide Mimic For The Active Site Of Cytochrome C Oxidase
Max E. Mahoney, Olof Einarsdottir, and Joseph P. Konopelski

PO-98
On The Mechanism Of 7-endo Selective Radical Cyclization Reaction To Give 2-Benzazepines And Exploration Of Their Biological Activity
Yuriko Ishihara, Masahiro So, Takahiro Hayashi, Makoto Inui, and Akio Kamimura

PO-99
Synthesis And Cytotoxic Activity Of Siliacycloalkyl Substituted Furans
Luba Ignatovich, Velta Muravenko, Ilze Sleiksha, Irina Shestakova, and Edmunds Lukevics

PO-100
Synthesis of Two Diastereomers of Monohydroxylated Metabolites Of BMS-562086
Jung-Hui Sun, Sarah C. Traeger, Robert R. Espina, Michael A. Witkus, Dauh-Rurng Wu, John D. DiMarco, Peggy Liu-Kreyche, Lian Zhou, Ramaswamy A. Iyer, Balu Balasubramanian, and Bang-Chi Chen

PO-101
A DOS Approach To Access A Full Stereochemical Matrix Of Complex Heterocycles Using SNAr As the Key Step: Solid-Phase Library Synthesis And Biological Evaluation
Jeremy Duvall, Baudouin Gerard, Haibo Liu, Jason T.Lowe, Tiffanie Murillo, Bhaumik Pandya, Byung-Chul Suh, Jingqiang Wei, Damian Young, and Lisa Marcaurelle

PO-102
Novel Dual Action Neuronal Nitric Oxide Synthase Inhibitors With 5-HT1D/1B Agonist Activity For The Treatment of Migraine Pain
Gabriela Mladenova, Subhash Annedi, Jailall Ramnauth, Joanne Speed, Paul Renton, Shawn Maddaford, Suman Rakhit, John Andrews, and Rob Medve

PO-103
Convenient Synthesis Of Oligonucleotides Bearing Novel Nucleobase Analogues By Post-Elongation Modification Method
Motoi Nakahara, Takeshi Kuboyama, Akhiro Izawa, Yoshiyuki Hari, Takeshi Imanishi, and Satoshi Obika

PO-104
The Effect Of Pyridinyl Nitrogen To Induce Chirality Organization Of Ferrocene-Dipeptide Bioconjugates
Toshiyuki Moriuchi, Takayoshi Nagai, Takashi Fujiwara, and Toshikazu Hirao

PO-105
Application of Enantioselective [2,3]-Wittig Rearrangement Construction Of Lignan Skeletons
Maria Kitamura, Yoshimi Hirokawa, Naoyoshi Maezaki

PO-106
Labelling Of 2’,5’-Oligoadenylates (2-5As) By Click Reaction
Takao Shiraishi, Yoshiaki Kitamura, Yoshihito Ueno, and Yukio Kitade

PO-107
Shape-Persistent Diethynylpyrene Macrocycles: Synthesis And Optoelectronic Properties
Gandikota Venkata Ramana, Matthew Curran, Simon Brake, Jay Duffet, and Graham J. Bodwell

PO-108
A Concise Approach To New Donor-Acceptor Xanthone-Carbazole Systems And Progress Toward Synthesis Of Cyclo-oligophenylenes
Anh-Thu Dang and Graham J. Bodwell

PO-109
A Paal-Knorr Approach To Lamellarins
Alfredo Vazquez, Armando Ramirez-Rodriguez, J. Manuel Mendez, Cristina Jimenez, and Fernando Leon

Wednesday August 5, 2009

Main Session (Salon A)

IL-12 9:00-9:30
New Asymmetric Methods for Heterocyclic Synthesis – Total Synthesis of Marinomycin A
P. Andrew Evans

PL-5 9:30-10:30
Synthetic studies of oxindole-containing natural products
John L. Wood (Winner of Katritzky Junior Award)

IL-13 11:00-11:30
Synthetic Study on Polyketide-Derived Polycyclic Natural Products
Keisuke Suzuki and Hiroshi Takikawa

PL-6 11:30-12:30
Chemical Synthesis in the Study of Biologically Active Natural Products
Samuel J. Danishefsky (Winner of ISHC Senior Award)

Thursday August 6, 2009

Main Session (Salon A)

PL-7 9:00-10:00
Synthetic Studies on Seemingly Simple Heterocyclic Natural Products
Tohru Fukuyama

IL-14 10:00-10:30
Epoxide-Opening Cascades
Timothy F. Jamison

PL-8 11:00-12:00
The use of functionalized ß-lactams as building blocks in heterocyclic chemistry
Matthias D’hooghe, Stijn Dekeukeleire and Erika Leemans Norbert De Kimpe

IL-15 12:00-12:30
Development of an Efficient Asymmetric Chemical Process for a Biologically Active Heterocycle
George A. Moniz

IL-16 1:30-2:00
The Role of 1,3-Dipolar Cycloaddition Reactions in the Design and Synthesis of Complex Heterocyclic Scaffolds with Anti-tumor/Anti-infective Activity
Anna Maria Almerico, Antonino Lauria & Gaetano Dattolo

OL-33 2:00-2:20
Synthesis of Impurities and/or Degradation Products of Zaleplon as an Integral Part of the API Development
Stanislav Radl, Michaela Blahovcova

OL-34 2:20-2:40
Radical Cyclization Routes to Benzimidazolequinones Containing Fused Aryl Rings: Access to a New Family of Bioreductive Anti-Tumor Agents
Eoin Moriarty , Fawaz Aldabbagh

OL-35 2:40-3:00
The Design, Synthesis, and Evaluation of Novel Substituted 5-Hydroxycoumarin and Pyrano-Coumarin Derivatives Exhibiting High Antiproliferative Activity
Gong-Chang Zeng, Wei-Wei Mao, Ting-Ting Wang, He-Ping Zeng

OL-36 3:30-3:50
NHC-Copper(I)-Catalyzed Asymmetric Allylic Substitution With Aryl Grignard Reagents
Khalid B.Selim, Yasumasa Matsumoto, Ken-ichi Yamada, & Kiyoshi Tomioka

OL-37 3:50-4:10
Structure-Activity Studies in Assessing the Surface Activity of Fluorous 1,2,3-Triazoles and Tetrazoles
Roger W. Read, Xiaobei Wang

OL-38 4:10-4:30
Structure-Based Design, Synthesis and Biological Evaluation for a Novel Series of Quercetin Diacylglucosides as a Potent Anti-MRSA agents.
Abugafar Md. Lokman Hossion, Nao Otsuka, Rafiya Khan Kandahary, Tomofusa Tsuchiya, Yoshito Zamami, & Kenji Sasaki

OL-39 4:30-4:50
Medical Materials For Early Finding and Curing Tumors: Synthesis and Evaluation of Deoxybromo-Phospha Sugars For Anti-Tumor Agents
Junko Yamashita, Mitsuji Yamashita, Manabu Yamada, Taishi Niimi, Michio fujie, Kazuhide Asai, Takuya Suyama, Maddali Kasthuraiah Reddy, & Satoki Nakamura

Session 1 (Salon C)

IL-17 1:30-2:00
Stereoselective Synthesis of Chiral Aziridines
Helene Lebel

OL-40 1:30-2:00
3-Oxa-1-Azabicyclo[3.1.0]-Hexan-2-one As a Convenient Starting Scaffold for the Synthesis of Imidazolinones, Substituted Piperazines and Piperazino[1,2-e]Triazoles
Iwona Maciagiewicz, Fang Fang, George Acquaah-Harrison, Corrina Grost, Ryan J. Roble, Dennis Roberts, Stephen C. Bergmeier

OL-41 2:20-2:40
New Gas-Phase Cascade Reactions of Stablised Phosphorus Ylides Leading to Ring-Fused Indoles and to Quinolines
R. Alan Aitken, Lorna Murray

OL-42 2:40-3:00
One-Pot Multi-Step Protocols for Synthesis of Novel Heterocyclic Frameworks
Pushpa Pardasani, R.T.Pardasani, Rahul Joshi & Sonali Verma

OL-43 3:30-3:50
New Routes to Azetidine Derivatives via Two- and Three-Component Reactions With Congested 1-Azabicyclo[1.1.0]Butanes
Grzegorz Mloston

OL-44 3:50-4:10
Synthesis of Isonucleosides and Cyclobutane Nucleoside Analogues
Abdelaziz Ebead, Edward Lee-Ruff

OL-45 4:10-4:30
Synthesis of Benzotriazine and Aryl-Triazene Derivatives Starting with 2-Azidobenzonitrile Derivatives
Azadeh Nakhai, Birgitta Stensland, Per H. Svensson & Jan Bergman

Session 2 (Salon D)

IL-18 1:30-2:00
Nickel-Catalyzed Synthesis of Oxazoles via C-S Activation
James P. Stambuli

OL-46 2:00-2:20
Total Synthesis of (+)-Myxothiazols A and Z
Hiroyuki Akita

OL-47 2:20-2:40
Synthetic Studies on (+)-Nakadomarin A
Fuyuhiko Inagaki, Masahiko Kinebuchi, Naoki Miyakoshi, Shinji Kitagaki & Chisato Mukai

OL-48 2:40-3:00
Synthetic Studies on (+)-Manzamine A
Tatsuya Toma, Yoichi Kita, Toshiyuki Kan, Tohru Fukuyama

OL-49 3:30-3:50
Synthesis And Anti-HIV Activity of Caffeoyl 5-Dehydroquinic Acid Derivatives
Chao-Mei Ma, Takuya Kawahata, Masao Hattori, Toru Otake, Mohsen Daneshtalab & Lili Wang

OL-50 3:50-4:10
New Synthetic Approach to Xanthone Natural Products Using N-Heterocyclic Carbene Catalysis
Yumiko Suzuki, Yoshinori Fukuta, Shinya Ota, Yuki Ueda, Masayuki Sato

OL-51 4:10-4:30
Reactions of 3-Oxopyridazine Derivatives with Some Active Amino and Methylene Compounds
Mohamed A. Khalil

OL-52 4:30-4:50
The Vegetal Refining of Lignocellulose: A New Era For the Furanic Chemistry
Bouchra Benjelloun- Mlayah, Yves le Bigot, Joseph H. Banoub, & Michel Delmas

Friday August 7, 2009

Main Session (Salon A)

PL-9 9:00-10:00
Synthesis of Biological Active cADPR Mimics
Li-He Zhang

IL-19 10:00-10:30
Heterocycles from Cyclopropanes: Enabling Methods for the Total Synthesis of Alkaloids
Michael A. Kerr

PL-10 11:00-12:00
Total Synthesis as a Vehicle for Penetrating Biomechanistic Puzzles: Challenges in Natural Products Chemistry
Robert M. Williams

SL 12:00-12:20
100 Years of Houben-Weyl and Science of Synthesis – Why you should care.
Thomas Krimmer